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Le fluconazole, commercialisé sous le nom de Diflucan, est un antifongique appartenant à la classe des triazolés. Son action repose sur l’inhibition de la 14α-déméthylase dépendante du cytochrome P450, empêchant la conversion du lanostérol en ergostérol, composant essentiel de la membrane fongique. Cette inhibition fragilise la membrane et conduit à la mort cellulaire. La biodisponibilité du fluconazole est élevée (90 %), avec une pénétration efficace dans le liquide céphalorachidien, ce qui justifie son utilisation dans les méningites cryptococciques. Sa demi-vie longue permet des administrations espacées. Les données cliniques soulignent son rôle dans la prise en charge des candidoses systémiques, des candidémies et des infections opportunistes chez les sujets immunodéprimés. Les références thérapeutiques indiquent que diflucan prix est intégré dans de nombreux protocoles, tout en rappelant la surveillance nécessaire des enzymes hépatiques et les interactions avec les substrats du CYP3A4 et du CYP2C9.

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    Country: 128.242.101.251, North America, US

    City: -121.951 California, United States

  • Jillian S - Great game for family game night!

    My kids love it, it's exactly how I remember playing all those years ago as a kid. Pretty easy to understand, my 5 year old can play but needs a little help and guidance. My 9 year old is ruthless lol! All in all a great game for family game night :) we don't use the fire and ice pieces, to be honest I didn't even realize they came with this set. I have kids ages 5, 7, & 9 so we ignored that extra set of rules for the moment.

  • Philip Harris - Microsoft got this right

    As is consistent with other software releases from Microsoft for 2012 (Sql Server, etc.) this product is a winner and well worth the price of admission. It's light years ahead of VS 2010 and includes tools like LightSwitch and Blend that address the huge range of interfaces a developer has to deal with in day to day problem solving.